Message: | Description:
Tibolonis a synthetic hormone-type drug which is used mainly for hormone replacement therapy in post-menopausal women.
it helps restore hormonal balance in the body.
When estrogen levels are low tissues can slowly degenerate, as is experienced during menopause. In addition, low levels of estrogen can cause distressing symptoms such as hot flushes, night sweats, mood swings, reduced sex drive and vaginal dryness.Tibolon is broken down into three compounds which act in a similar way to the natural estrogen and progesterone found in the body. It restores plasma endorphin level in post-menopausal women and acts centrally to affect the thermo-regulatory system.
Tibolone
Product name: Tibolone
Synonym: TIBOLONE;LIVIELLA;LIVIAL;5(10)-ESTREN-7-ALPHA-METHYL-17-ALPHA-ETHYNYL-17-BETA-OL-3-ONE;(7A,17A)-17-HYDROXY-7-METHYL-19-NORPREGN-5(10)-EN-20-YL-3-ONE;17-hydroxy-7alpha-methyl-19-norpregn-5(10)-en-20-yn-3-one;17ALPHA-HYDROXY-7ALPHA-METHYL-19-NORPREGN-5(10)-EN-20-YN-3-ONE;19-NORPREGN-5(10)-EN-20-YN-3-ONE,17-HYDROXY-7-METHYL-, (7A,17A)-
CAS Registry Number: 5630-53-5
Molecular Formula: C21H28O2
Molecular Weight: 312.45
Assay: 99% min.
Packing: 1kg/foil bag.
Delivery: Express courier
Usage: pharmaceutical material, Steroid hormone, Anabolin. A synthetic steroid with weak estrogenic, androgenic and progestogenic activity. A pharamceutical used in the treatment of menopausal syndrome.
Applications:
In itself Tibolon has no biological activity; the effects are produced mainly by the results of the activity of its metabolites on various tissues. After administration, it is quickly metabolized into 3α-hydroxytibolon and 3ß-hydroxytibolon compounds, which are also present in an inactive, sulfated form. A third compound, the Δ4- isomer is formed from Tibolon directly or from the 3ß hydroxymetabolite.
Tibolon has estrogenic effects on bone and vaginal tissue. |